Emmanuel Theodorakis

Personal Home Page

http://www-chem.ucsd.edu/research/profile.cfm?cid=C02377

Articles in Scholarly Journals [Incomplete List]

  1. Chalcogen-Substituted Benzo-1,4-quinones
    ChemInform, vol. 38, no. 36, 2007
  2. Nitrogen- and Phosphorus-Substituted Benzo-1,4-quinones
    ChemInform, vol. 38, no. 39, 2007
  3. Studies on the Synthesis ofSchisandraceae Natural Products: Exploring a Cyclopropylcarbinol Ring Expansion Strategy
    European Journal of Organic Chemistry, vol. 2007, no. 25, pp. 4193–4196, 2007
  4. Trifunctional norrisolide probes for the study of Golgi vesiculation
    Bioorganic & Medicinal Chemistry Letters, vol. 17, no. 2, pp. 320–325, 2007
  5. Synthesis and use of an in-solution ratiometric fluorescent viscosity sensor
    Nature Protocols, vol. 2, no. 1, Article ID nprot.2006.455, 9 pages, 2007
  6. Synthesis and evaluation of caged Garcinia xanthones
    Organic & Biomolecular Chemistry, vol. 5, no. 3, p. 494, 2007
  7. Molecular rotors?fluorescent biosensors for viscosity and flow
    Organic & Biomolecular Chemistry, vol. 5, no. 11, p. 1669, 2007
  8. Selective Activation of Liver X Receptors by Acanthoic Acid-Related Diterpenes
    Molecular Pharmacology, vol. 71, no. 6, pp. 1545–1553, 2007
  9. Optical fiber-based fluorescent viscosity sensor
    Optics Letters, vol. 31, no. 17, p. 2529, 2006
  10. Journal of the American Chemical Society, vol. 128, no. 2, pp. 398–399, 2006
  11. Journal of the American Chemical Society, vol. 128, no. 13, pp. 4190–4191, 2006
  12. Nature-inspired approaches to chemical synthesis
    Tetrahedron, vol. 62, no. 22, pp. 5169–5169, 2006
  13. A Central Strategy for Converting Natural Products into Fluorescent Probes
    ChemBioChem, vol. 7, no. 3, pp. 409–416, 2006
  14. Norrisolide: Total Synthesis and Related Studies
    Chemistry - A European Journal, vol. 11, no. 24, pp. 7175–7190, 2005
  15. A New Family of Synthetic Diterpenes that Regulates Cytokine Synthesis by Inhibiting I?B? Phosphorylation
    ChemBioChem, vol. 6, no. 1, pp. 133–144, 2005
  16. Quinone Sesquiterpenes: A Challenge for the Development of a New Synthetic Methodology
    ChemInform, vol. 36, no. 42, 2005
  17. Synthesis and evaluation of 6-hydroxy-7-methoxy-4-chromanone- and chroman-2-carboxamides as antioxidants
    Bioorganic & Medicinal Chemistry Letters, vol. 15, no. 11, pp. 2745–2748, 2005
  18. Effects of solvent polarity and solvent viscosity on the fluorescent properties of molecular rotors and related probes
    Bioorganic Chemistry, vol. 33, no. 6, pp. 415–425, 2005
  19. Synthetic studies toward the zoanthamine alkaloids: synthesis of the fully functionalized BC ring motif
    Tetrahedron Letters, vol. 46, no. 32, pp. 5281–5284, 2005
  20. Sensing of Flow and Shear Stress Using Fluorescent Molecular Rotors
    Sensor Letters, vol. 3, no. 1, pp. 42–48, 2005
  21. HIF-1  expression regulates the bactericidal capacity of phagocytes
    Journal of Clinical Investigation, vol. 115, no. 7, pp. 1806–1815, 2005
  22. Synthesis of Fused Tetrahydrofuran-?-lactone Motifs via One-Pot Ring Expansion of Cyclopropane Rings
    Synthetic Communications, vol. 34, no. 11, pp. 1951–1965, 2004
  23. 3,3-Oxybis(dimethoxytrityl chloride) (O-DMTCl): synthesis and applications of a novel bifunctional protecting group
    Bioorganic & Medicinal Chemistry Letters, vol. 14, no. 12, pp. 3241–3244, 2004
  24. Fragmentation of Golgi membranes by norrisolide and designed analogues
    Bioorganic & Medicinal Chemistry Letters, vol. 14, no. 20, pp. 5035–5039, 2004
  25. Synthesis and in vitro antitumor activity of phthalimide-based polymers containing camptothecin
    European Polymer Journal, vol. 40, no. 7, pp. 1291–1296, 2004
  26. Synthesis of (+)- and ($minus;)-isocarvone
    Tetrahedron Letters, vol. 45, no. 26, pp. 5039–5041, 2004
  27. Stereoselective Total Synthesis of (-)-Borrelidin.
    ChemInform, vol. 35, no. 47, 2004
  28. Stereoselective Total Synthesis of (+)-Norrisolide
    Angewandte Chemie International Edition, vol. 43, no. 6, pp. 739–742, 2004
  29. Stereoselective Total Synthesis of (-)-Borrelidin
    Angewandte Chemie International Edition, vol. 43, no. 30, pp. 3947–3951, 2004
  30. Hydrophilic molecular rotor derivatives?synthesis and characterization
    Bioorganic Chemistry, vol. 32, no. 4, pp. 274–289, 2004
  31. Natural Product Synthesis Special Feature: Unified synthesis of caged Garcinia natural products based on a site-selective Claisen/Diels-Alder/Claisen rearrangement
    Proceedings of the National Academy of Sciences, vol. 101, no. 33, pp. 12030–12035, 2004
  32. Organic Letters, vol. 6, no. 6, pp. 941–944, 2004
  33. Organic Letters, vol. 5, no. 10, pp. 1617–1620, 2003
  34. Organic Letters, vol. 5, no. 9, pp. 1491–1494, 2003
  35. Novel synthesis of 2'-O-methylguanosine
    Bioorganic & Medicinal Chemistry Letters, vol. 13, no. 10, pp. 1631–1634, 2003
  36. Synthesis of a novel family of diterpenes and their evaluation as anti-inflammatory agents
    Bioorganic & Medicinal Chemistry Letters, vol. 13, no. 19, pp. 3217–3221, 2003
  37. Synthesis and antitumour activity of medium molecular weight phthalimide polymers of camptothecin
    Polymer International, vol. 52, no. 8, pp. 1339–1345, 2003
  38. Total synthesis of seco-lateriflorone
    Tetrahedron, vol. 59, no. 35, pp. 6873–6887, 2003
  39. Total synthesis of atroviridin
    Tetrahedron Letters, vol. 44, no. 16, pp. 3281–3284, 2003
  40. Synthesis and biological activity of medium molecular weight polymers of camptothecin
    European Polymer Journal, vol. 39, no. 2, pp. 367–374, 2003
  41. Biomimetic total synthesis of forbesione and desoxymorellin utilizing a tandem Claisen/Diels?Alder/Claisen rearrangementElectronic supplementary information (ESI) available: 1H and 13C NMR spectra for compounds 1, 3, 8 and 9. See http://www.rsc.org/suppdata/ob/b3/b311833a/
    Organic & Biomolecular Chemistry, vol. 1, no. 24, p. 4418, 2003
  42. MDPSCL2: A New Protecting Group for Chemoselective Synthesis of 2'-O-Alkylated Guanosines
    Nucleosides, Nucleotides & Nucleic Acids, vol. 22, no. 5-8, pp. 583–587, 2003
  43. Stereoselective synthesis of the fully functionalized core fragment of terpentecin
    Tetrahedron Letters, vol. 43, no. 50, pp. 9019–9022, 2002
  44. Synthesis and biological activity of phthalimide-based polymers containing 5-fluorouracil
    Polymer International, vol. 51, no. 7, pp. 569–576, 2002
  45. Phospholipid-Bound Molecular Rotors: Synthesis and Characterization
    Bioorganic & Medicinal Chemistry, vol. 10, no. 11, pp. 3627–3636, 2002
  46. Journal of the American Chemical Society, vol. 124, no. 41, pp. 12261–12267, 2002
  47. The Journal of Organic Chemistry, vol. 67, no. 22, pp. 7887–7889, 2002
  48. Organic Letters, vol. 4, no. 6, pp. 909–912, 2002
  49. Organic Letters, vol. 4, no. 5, pp. 819–822, 2002
  50. The Journal of Organic Chemistry, vol. 66, no. 26, pp. 8843–8853, 2001
  51. Investigation of the biological mode of action of clerocidin using whole cell assays
    Bioorganic & Medicinal Chemistry, vol. 9, no. 6, pp. 1365–1370, 2001
  52. New fluorescent probes for the measurement of cell membrane viscosity
    Chemistry & Biology, vol. 8, no. 2, pp. 123–131, 2001
  53. Synthesis and biological activity of medium range molecular weight polymers containingexo-3,6-epoxy-1,2,3,6-tetrahydrophthalimidocaproic acid
    Polymer International, vol. 50, no. 9, pp. 1010–1015, 2001
  54. Stereoselective Total Synthesis of Reveromycin B and C19-epi-Reveromycin B
    Chemistry - A European Journal, vol. 6, no. 11, pp. 1987–2001, 2000
  55. Organic Letters, vol. 2, no. 14, pp. 2073–2076, 2000
  56. Organic Letters, vol. 2, no. 2, pp. 207–210, 2000
  57. Organic Letters, vol. 1, no. 8, pp. 1295–1297, 1999
  58. Design, synthesis, and evaluation of N-aroyloxy-2-thiopyridones as DNA photocleaving reagents
    Bioorganic & Medicinal Chemistry, vol. 7, no. 5, pp. 727–736, 1999
  59. Journal of the American Chemical Society, vol. 121, no. 2, pp. 456–457, 1999
  60. Enantioselective Total Synthesis of Avarol and Avarone
    Angewandte Chemie International Edition, vol. 38, no. 20, pp. 3089–3091, 1999
  61. On the mechanism of photo-induced nucleic acid cleavage using -aroyloxy-2-thiopyridones
    Tetrahedron Letters, vol. 39, no. 21, pp. 3383–3386, 1998
  62. Journal of Organic Chemistry, vol. 63, no. 20, pp. 6774–6775, 1998
  63. Photochemical cleavage of duplex DNA by N-benzoyloxy-2-thiopyridone linked to 9-aminoacridine
    Chemical Communications, no. 15, pp. 1463–1464, 1997
  64. Sequence-selective carbohydrate-DNA interaction: Dimeric and monomeric forms of the calicheamicin oligosaccharide interfere with transcription factor function
    Proceedings of the National Academy of Sciences, vol. 93, no. 2, pp. 940–944, 1996
  65. N-aroyloxy-2-thiopyridones as efficient oxygen-radical generators: novel time-controlled DNA photocleaving reagents
    Chemical Communications, no. 16, p. 1927, 1996
  66. Chemistry and biology of selected natural products
    Pure and Applied Chemistry, vol. 68, no. 11, pp. 2129–2136, 1996
  67. Journal of the American Chemical Society, vol. 117, no. 3, pp. 1171–1172, 1995
  68. Journal of the American Chemical Society, vol. 117, no. 3, pp. 1173–1174, 1995
  69. Journal of the American Chemical Society, vol. 117, no. 41, pp. 10227–10238, 1995
  70. Journal of the American Chemical Society, vol. 117, no. 41, pp. 10239–10251, 1995
  71. Journal of the American Chemical Society, vol. 117, no. 41, pp. 10252–10263, 1995
  72. The relationship of brevetoxin ?length? and A-ring functionality to binding and activity in neuronal sodium channels
    Chemistry & Biology, vol. 2, no. 8, pp. 533–541, 1995
  73. Synthetic calicheamicin mimics with novel initiation mechanisms: DNA cleavage, cytotoxicity, and apoptosis
    Chemistry & Biology, vol. 1, no. 1, pp. 57–66, 1994
  74. A convenient and high yielding procedure for the preparation of isoselenocyanates. Synthesis and reactivity of ?-alkylselenocarbamates.
    Tetrahedron, vol. 50, no. 37, pp. 639–654, 1994
  75. Journal of the American Chemical Society, vol. 116, no. 20, pp. 9371–9372, 1994
  76. Journal of the American Chemical Society, vol. 115, no. 18, pp. 8050–8059, 1993
  77. Journal of the American Chemical Society, vol. 114, no. 14, pp. 5904–5905, 1992
  78. The invention of radical reactions. Part XXIII new reactions: Nitrile and thiocyanate transfer to carbon radicals from sulfonyl cyanides and sulfonyl isothiocyanates.
    Tetrahedron, vol. 48, no. 13, pp. 2613–2626, 1992
  79. O-Sulfinylation of alcohols with methanesulfonyl cyanide or p-toluenesulfonyl cyanide.
    Tetrahedron, vol. 47, no. 44, pp. 9167–9178, 1991
  80. O-sulfinylation with methanesulfonyl cyanide or p-toluenesulfonyl cyanide and DBU.
    Tetrahedron Letters, vol. 32, no. 23, pp. 2585–2588, 1991
  81. Radical nitrile transfer with methanesulfonyl cyanide or p-toluenesulfonyl cyanide to carbon radicals generated from the acyl derivatives of N-hydroxy-2-thiopyridone
    Tetrahedron Letters, vol. 32, no. 28, pp. 3321–3324, 1991
  82. Asymmetric Synthesis XXIII.1 A 100% cis Diastereoselectivity in the SYnthesis of Enantiomerically Pure 2,6-Dialkylpiperidines
    Synthetic Communications, vol. 21, no. 4, pp. 521–529, 1991