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Larry C. Wienkers
Articles in Scholarly Journals [Incomplete List]
CYP2C9 Protein Interactions with Cytochrome b5: Effects on the Coupling of Catalysis
Drug Metabolism and Disposition, vol. 35, no. 7, pp. 1174–1181, 2007
Chemical Research in Toxicology, vol. 19, no. 12, pp. 1650–1659, 2006
Mechanism of Inactivation of Human Cytochrome P450 2B6 by Phencyclidine
Drug Metabolism and Disposition, vol. 34, no. 9, pp. 1523–1529, 2006
The in Vitro Drug Interaction Potential of Dietary Supplements Containing Multiple Herbal Components
Drug Metabolism and Disposition, vol. 35, no. 2, pp. 185–188, 2006
Predicting in vivo drug interactions from in vitro drug discovery data
Nature Reviews Drug Discovery, vol. 4, no. 10, Article ID nrd1851, 8 pages, 2005
Catalytic turnover of pyrene by CYP3A4: Evidence that cytochrome directly induces positive cooperativity
Archives of Biochemistry and Biophysics, 2005
Chemical Research in Toxicology, vol. 17, no. 2, pp. 174–184, 2004
IN VITRO METABOLISM OF CLINDAMYCIN IN HUMAN LIVER AND INTESTINAL MICROSOMES
Drug Metabolism and Disposition, vol. 31, no. 7, pp. 878–887, 2003
Activation of cytochrome P450 2C9-mediated metabolism: mechanistic evidence in support of kinetic observations
Archives of Biochemistry and Biophysics, vol. 410, no. 1, pp. 16–24, 2003
Effect of carbonate anion on cytochrome P450 2D6-mediated metabolism in vitro: the potential role of multiple oxygenating species
Archives of Biochemistry and Biophysics, vol. 417, no. 2, pp. 165–175, 2003
Journal of Medicinal Chemistry, vol. 46, no. 2, pp. 284–302, 2003
Chemical Research in Toxicology, vol. 16, no. 4, pp. 450–459, 2003
Characterization of bropirimine O -glucuronidation in human liver microsomes
Xenobiotica, vol. 33, no. 10, pp. 999–1011, 2003
Pyrene·Pyrene Complexes at the Active Site of Cytochrome P450 3A4: Evidence for a Multiple Substrate Binding Site
Journal of the American Chemical Society, vol. 124, no. 40, pp. 11866–11867, 2002
Factors confounding the successful extrapolation of in vitro CYP3A inhibition information to the in vivo condition
European Journal of Pharmaceutical Sciences, vol. 15, no. 3, pp. 239–242, 2002
Multiple Cytochrome P450 Enzymes Responsible for the Oxidative Metabolism of the Substituted (S)-3-Phenylpiperidine, (S,S)-3-[3-(Methylsulfonyl)phenyl]-1-propylpiperidine Hydrochloride, in Human Liver Microsomes
Drug Metabolism and Disposition, vol. 30, no. 12, pp. 1372–1377, 2002
Problems associated with in vitro assessment of drug inhibition of CYP3A4 and other P-450 enzymes and its impact on drug discovery
Journal of Pharmacological and Toxicological Methods, vol. 45, no. 1, pp. 79–84, 2001
Covalent Alteration of the CYP3A4 Active Site: Evidence for Multiple Substrate Binding Domains
Archives of Biochemistry and Biophysics, vol. 391, no. 1, pp. 49–55, 2001
Identification of cytochrome P4503A as the major subfamily responsible for the metabolism of roquinimex in man
Xenobiotica, vol. 30, no. 9, pp. 905–914, 2000
Chemical Research in Toxicology, vol. 13, no. 4, pp. 262–270, 2000
In vitro metabolic transformations of 2,4- dipyrrolidinylp yrimidine : a chemical probe for P450-mediated oxidation of tirilazad mesylate
Xenobiotica, vol. 27, no. 11, pp. 1131–1145, 1997