Sweetening Pharmaceutical Radiochemistry by ¹⁸F-Fluoroglycosylation: A Short Review

Scheme 1

General reaction scheme for [¹⁸F]fluoroglycosylation via CuAAC using 2-deoxy-2-[¹⁸F]fluoroglucopyranosyl azide 3, starting from the β-mannosyl azide 1.