Sweetening Pharmaceutical Radiochemistry by ¹⁸F-Fluoroglycosylation: A Short Review

Table 3

¹⁸F-Glycoconjugates synthesized by miscellaneous ¹⁸F-fluoroglycosylation.

Structure	Conjugation	Target	Reference
	Enzymatic glycosylation	Glycosyltransferases	[39, 40]
	Enzymatic glycosylation	𝛽-Galactosidase/LacZ gene	[41]
	Enzymatic glycosylation	GCase	[42]
	Lewis acid promoted N-glycosylation	Hypoxia	[43]
	Thiol-selective S-glycosylation	Integrin 𝛼𝑣𝛽3	[44]
	Thionation + site selective conjugation	Cys-containing proteins	[45]
		Breast cancer cells	[46, 47]