|
Target/mechanism | Imaging agent | Disease/microorganism (study type) |
|
| Inflammation | |
|
P-selectin | 68GaGa-Fucoidan | Atherosclerotic plaques (preclinical [44]) |
|
Anti-CD163 | 68GaGa-anti-CD163-antibody | Acute collagen-induced arthritis (preclinical [45]) |
|
Integrins | 68GaGa-PRGD2 | Rheumatoid arthritis (clinical [46]) |
|
Integrins | 68GaGa-NOTA-c(RGDyK) 68GaGa-NODAGA-RGD 68GaGa-TRAP-(RGD)3 68Ga-DOTA-E-c (RGDfK)2 | Myocardial infarction (preclinical [47–51]) |
|
Integrins | 68GaGa-NODAGA-RGD | Atherosclerotic plaques (preclinical [52]) |
|
VAP-1 | 68GaGa-Siglec | Synovial inflammation; inflammatory lung injury; atherosclerotic lesions; skin/muscle inflammation (preclinical [53–56]) |
|
VAP-1 | 68GaGa-DOTAVAP-P1, 68GaGa-DOTAVAP-PEG-P1 | Skin/muscle inflammation (preclinical [57]) |
|
CXCR4 | 68GaGa-pentixafor | Ischemic heart; atherosclerotic plaques (clinical [58, 59]) |
|
FR | 68GaGa-DOTA-PEG-FA 68GaGa-DOTA-folate | Inflammation/implant (preclinical [60, 61]) |
|
SSTR | 68GaGa-DOTA-TOC | Sarcoidosis, idiopathic pulmonary fibrosis, Graves’ disease, Hashimoto’s disease, coronary artery plaque, atherosclerotic inflammation (clinical [62–65]) |
|
Mannose receptors | 68GaGa-NOTA-MSA | Myocarditis (preclinical [66]) |
|
Aβ plaques | 68Ga-labelled styrylpyridines, benzofuran, curcumin | Neuroinflammation, Alzheimer’s disease (preclinical [67–69]) |
|
| Infection | |
|
Antibiotics/inhibitor | 68GaGa-ciprofloxacin | Staphylococcus aureus (preclinical [70]) |
|
Antimicrobial/membrane | 68GaGa-NOTA-UBI29-41 68GaGa-NOTA-UBI30-41 | Staphylococcus aureus (preclinical [71, 72]) |
|
Antimicrobial/membrane | 68GaGa-DOTA-TBIA101 | E. coli (preclinical [73, 74]) |
|
Antimicrobial/membrane | 68GaGa-GF-17 and 68GaGa-RAWVAWR-NH2 | E. coli and S. aureus (preclinical [75]) |
|
Siderophores | 68GaGa-TAFC, 68GaGa-FC, 68GaGa-FOXE | Invasive pulmonary aspergillosis (preclinical [15, 16, 76]) |
|
Leukocytes | 68GaGa-citrate | Osteomyelitis, diskitis, intra-abdominal infection, tuberculosis, interstitial nephritis (clinical [18, 19, 77–80]) |
|
Leukocytes | 68GaGa-Apo-transferrin | Staphylococcus aureus (preclinical [14]) |
|