International Journal of Experimental Diabetes Research
Volume 3 (2002), Issue 3, Pages 163-169
doi:10.1080/15604280214280

Fasting Decreases the Content of D-Chiroinositol in Human Skeletal Muscle

Pavel N. Shashkin,1 Laura C. Huang,2 Joseph Larner,2 George E. Vandenhoff,2 and Abram Katz3

1Department of Internal Medicine, University of Virginia Charlottesville, Charlottesville, Virginia, USA
2Department of Pharmacology, University of Virginia Charlottesville, Charlottesville, Virginia, USA
3Department of Physiology and Pharmacology, Karolinska Institutet, Stockholm 171 77 , Sweden

Received 28 October 2001; Accepted 21 February 2002

Copyright © 2002 Pavel N. Shashkin et al. This is an open access article distributed under the Creative Commons Attribution License, which permits unrestricted use, distribution, and reproduction in any medium, provided the original work is properly cited.

Abstract

Two classes of inositol phosphoglycans have been implicated as second messengers of insulin, one that activates pyruvate dehydrogenase and contains D-chiroinositol, and one that inhibits cyclic AMP–dependent protein kinase and contains myoinositol. We examined the effects of a 3-day fast on muscle contents of inositols in healthy humans. An oral glucose tolerance test was performed and a biopsy was obtained from the quadriceps femoris muscle after an overnight fast and after a 72-hour fast. The 72-hour fast significantly increased plasma glucose (1.5- to 2-fold) and insulin (2- to 4-fold) after glucose ingestion versus the values after the overnight fast, indicating the manifestation of peripheral insulin resistance. The 72-hour fast resulted in an ∼20% decrease in the muscle content of D-chiroinositol (P < 0.02), but no change in the myoinositol content. These data demonstrate that fasting specifically decreases the muscle content of D-chiroinositol in human muscle and this may contribute to the finding that insulin-mediated activation of pyruvate dehydrogenase is attenuated after short-term starvation.