Table 1:
One-pot synthesis of benzo[
b
]1,8-naphthyridines.
Entry
R
R
1
R
2
𝑃
𝑟
o
d
u
c
t
a
Yield
(
%
)
b
1
H
H
H
4a
93
2
CH
3
H
H
4b
95
3
OCH
3
H
H
4c
95
4
Cl
H
H
4d
97
5
CH
3
CH
3
H
4e
93
6
H
H
CH
3
4f
95
7
H
H
OCH
3
4g
96
8
H
H
Cl
4h
96
a
A
l
l
the products were characterised by IR,
1
H
NMR, and mass spectra.
b
Y
i
e
l
d
s
of isolated products.