Benzo[1,5]thiazepine: Synthesis, Reactions, Spectroscopy, and Applications
Scheme 46
Reaction of 2-(bromomethyl)-1-sulfonylaziridines with 2-aminothiophenol in THF in the presence of K2CO3: A regio- and stereocontrolled synthesis of trans-2-phenyl- and trans-4-(phenyl or propyl)-3-sulfonamido-2,3,4,5-tetrahydro-1,5-benzothiazepines.
