Review Article

Emerging Therapeutic Strategies for Targeting Chronic Myeloid Leukemia Stem Cells

Table 1

Summary of the tyrosine kinase inhibitors and their effects on T315I.

TKIOriginally termedTKI generation Acts on T315I

ImatinibSTI571First No
Dasatinib BMS-354825Second No
Nilotinib AMN107Second No
Bosutinib SKI-606Second No
Ponatinib AP24534Third Yes