Review Article

Plasma Membrane Transporters in Modern Liver Pharmacology

Table 3

Identified potential substrates of hepatic forms of CNTs, ENTs, and PEPTs with pharmacological interest.

CNT1-3ENT1-3PEPT1-2

SubstratesAdenine5-Aminolevulinic acid
Amoxicillin
Ampicillin
AdenosineAdenosineBestatin
Benzamide ribosideCefadroxil
CladribineCladribineCefixime
ClofarabinClofarabineCeftibuten
CytarabineCephalexin
CytidineCytidineCephradine
DidanosineGlycylsarcosine
FialuridineFialuridineL-Kyotorphin
FludarabineFludarabine
5-Fluorouridine
Formycin
GemcitabineGemcitabine
Guanine
GuanosineGuanosine
Hypoxanthine
6-Mercaptopurine
InosineInosine
RibavirinRibavirin
Stavudine
6-Thioguanine
ThymidineThymidine
TiazofurinTiazofurin
UridineUridine
Zalcitabine
ZebularineZebularine
ZidovudineZidovudine