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| | Compd. | –R | values | IC90 (g/mL) | CC50 (g/mL) VERO | SI |
| | 1a | HCO | −1.1502 | <0.20 | >37.43 | >187.1 | | b | CH3CO | −1.2042 | <0.20 | >41.64 | >208.2 | | c | CF3CO | −0.0952 | 0.281 | >44.23 | >156.8 | | d | CHCl2CO | 0.1218 | <0.20 | >45.72 | >228.6 | | e | CH3CH2CO | −0.6752 | 0.334 | >40.24 | >120.4 | | f | CH3CH2OCO | 0.9748 | 0.422 | >41.84 | >98.91 | | g | (CH3)2CHCO | −0.3662 | 0.283 | >41.64 | >146.6 | | h | (CH3)3COCO | 1.6828 | <0.20 | >44.64 | >223.2 | | i | CH3(CH2)4CO | 0.9118 | <0.20 | >44.45 | >222.2 | | j | cyclohexanoyl | 0.8268 | 2.095 | >45.65 | >21.79 | | k | CH3(CH2)5CO | 1.4408 | <0.20 | >45.85 | >229.2 | | l | CH3(CH2)6CO | 1.9698 | <0.20 | >47.25 | >236.2 | | m | CH3(CH2)7CO | 2.4988 | <0.20 | >48.65 | >243.2 | | n | CH3(CH2)8CO | 3.0278 | <0.20 | >50.06 | >250.3 | | o | CH3(CH2)9CO | 3.5568 | <0.20 | >51.46 | >257.3 | | p |  | 1.7208 | <0.20 | >48.25 | >241.2 | | PH-27 |  | 0.6308 | 0.466 | >34.73 | >74.53 | | LZD |  | 0.5321 | <0.20 | >33.73 | >168.6 | | INH |  | −0.668 | 0.034 | >100 | >2941 |
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