Research Article

Evaluation of Novel 3-Hydroxyflavone Analogues as HDAC Inhibitors against Colorectal Cancer

Table 2

Whole cell HDAC enzyme inhibition assay.

Sl. no.CompoundHDAC inhibition IC50 (µM ± SEM)

1QMJ-11023.1 ± 5.2
2QMJ-2181.7 ± 22.04
3QMJ-31124 ± 6.2
4QMJ-41011.2 ± 3.4
5QMJ-570.2 ± 4.3
6QMJ-6984.2 ± 2.5
7Quercetin167.8 ± 6.9
8SAHA1.2 ± 0.1

The values are expressed as mean ± SEM of three experiments.