Research Article

Targeted Tumor Therapy with Radiolabeled DNA Intercalator: A Possibility? Preclinical Investigations with 177Lu-Acridine

Table 1

Variation of radiolabeling yield of 177Lu-acridine complex with incubation temperature.

Incubation temperature (°C)% Radiolabeling yield

Room temperature (27)
50
100

Radiolabeling studies were carried out using 1.5 mg/mL acridine-DOTA conjugate at pH 5 for 45 min. Experiments were done in triplicate.