| Rank | Western medications () | Chinese herbal medications () | Products (compound) | | % | Products (Chinese name) | Ingredients (Latin name) | | % |
| 1 | Cyproterone acetate | 70 | 4.6 | Bai Mao Gen | Rhizoma Imperatae Cylindricae | 40 | 3.5 |
| 2 | Tamsulosin | 63 | 4.1 | Ma Zi Ren Wan | Fructus Cannabis, Radix Paeoniae, Fructus Aurantii Immaturus, Radix et Rhizoma Rhei, Cortex Magnoliae Officinalis, Semen Armeniaccae Amarum | 35 | 3.1 |
| 3 | Magnesium oxide | 60 | 3.9 | Da Huang | Radix et Rhizoma Rhei | 31 | 2.7 | | | | | Sheng Di Huang | Radix Rehmanniae | 31 | 2.7 |
| 4 | Imipramine | 50 | 3.3 | Zuo Gui Wan | Radix Rehmanniae, Glutinosae Conquitae, Fructus Corni Officinalis, Fructus Lycii, Colla Cornus Cervi, Semen Cuscutae Chinensis, Radix Dioscoreae Oppositae, Colla Carapacis et Plastri Testudinis, Radix Achyranthis Bidentatae | 29 | 2.5 |
| 5 | Terazosin | 49 | 3.2 | Niu Xi | Radix Achyranthis Bidentatae | 28 | 2.4 |
| 6 | Leuprolide acetate | 43 | 2.8 | Che Qian Zi | Semen Plantaginis | 27 | 2.4 |
| 7 | Tolterodine L-tartrate | 40 | 2.6 | Yu Mi Xu | Stigma Maydis | 26 | 2.3 | | | | | Zhu Ru | Caulis Bambusae in Taeniis | 26 | 2.3 |
| 8 | Doxazosin | 34 | 2.2 | Gui Zhi Fu Ling Wan | Ramulus Cinnamomi, Sclerotium Poriae Cocos, Cortex Moutan Radicis, Semen Persicae, Radix Paeoniae Rubra | 26 | 2.3 |
| 9 | Sennoside | 30 | 2.0 | Gui Lu Er Xian Jiao | Colla Carapacis et Plastri Testudinis, Colla Cornus Cervi, Fructus Lycii, Radix Ginseng | 23 | 2.0 |
| 10 | Alfuzosin | 29 | 1.9 | Shu Jing Huo Xue Tang | Radix Glycyrrhizae, Radix Angelicae Sinensis, Radix Paeoniae Alba, Radix Rehmanniae, Rhizoma Atractylodis, Radix Cyathulae, Pericarpium Citri Reticulatae, Semen Persicae, Radix et Rhizoma Clematidis, Rhizoma Chuanxiong, Radix Stephaniae Tetrandrae, Rhizoma et Radix Notopterygii, Radix Saposhnikoviae, Radix Angelicae Dahuricae, Gelatinum Plastri Testudinis, Poria, Rhizoma Zingiberis Recens | 22 | 1.9 |
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