Review Article

The Chemical Constituents and Pharmacological Actions of Cordyceps sinensis

Table 1

Chemical constituents and their corresponding pharmacological actions of C. sinensis.

Chemical constituents of C. sinensis Pharmacological effectsReferences

CordycepinAnti-inflammatory effect[17, 2130]
Analgesic effect
Stimulates steroidogenesis
Enhances immunity
Antitumor activity
Antibacteria, antivirus, and insecticidal activities

AdenosineAnticonvulsant activity [20, 3146]
Inhibits cancer cell growth
Anti-inflammatory effect

EPSFImmunomodulatory effect[6065]
Antitumour effect
Antioxidant effect

APSAntioxidant effect[6669]
Immunomodulatory effects

CPS-1Antioxidant effect[70, 71]

CPS-2Inhibits cell proliferation[72, 73]

MannoglucanCytotoxicity activity[74]

CME-1Antioxidant effect[75]

CordyglucansAntitumour effect[76]

CS-F10Hypoglycemic activity[55, 77]

CordysinocanInduces cell proliferation[77]

ErgosterolCytotoxicity[7883]
Antimicrobial activity

H1-AImmunoregulation[8486]

CSDNaseHydrolyzes DNA[89, 90]
Nucleolytic properties

CSPFibrinolytic activity[91]

CordyminAntidiabetic[9395]

TryptophanSedative hypnotic effect[98]

Cordycepic acidTreating liver fibrosis diuretic[99103]
Improving the plasma osmotic pressure
Anti-free radical

Monosaccharide saponinsAntitumor activity[104]