Urotensin-II Ligands: An Overview from Peptide to Nonpeptide Structures

Table 1

Name	Peptide sequence
PRL-2903	H-4Fpa-c[Cys-Pal-DTrp-Lys-Tle-Cys]-Nal-NH2
SB-710411	H-Cpa-c[DCys-Pal-DTrp-Lys-Val-Cys]-Cpa-NH2
BIM-23127	H-D(2′)Nal-c[Cys-Tyr-DTrp-Orn-Val-Cys]-(2′)Nal-NH2
BIM-23042	H-DNal-c[Cys-Tyr-DTrp-Lys-Val-Cys]-(2′)Nal-NH2
[Orn^8]U-II	H-Glu-Thr-Pro-Asp-c[Cys-Phe-Trp-Orn-Tyr-Cys]-Val-OH
P5U	H-Asp-c[Pen-Phe-Trp-Orn-Tyr-Cys]-Val-OH
Urantide	H-Asp-c[Pen-Phe-DTrp-Orn-Tyr-Cys]-Val-OH
UFP-803	H-Asp-c[Pen-Phe-DTrp-Dab-Tyr-Cys]-Val-OH
URP	H-Ala-c[Cys-Phe-Trp-Lys-Tyr-Cys]-Val-OH
Urocontrin	H-Bip-c[Cys-Bip-Trp-Lys-Tyr-Cys]-Val-OH
GSK248451	H-Cin-c[DCys-Pal-DTrp-Orn-Val-Cys]-His-NH2