Research Article
Utilization of Boron Compounds for the Modification of Suberoyl Anilide Hydroxamic Acid as Inhibitor of Histone Deacetylase Class II Homo sapiens
Table 2
Catalytic site of HDAC class II Homo sapiens enzyme.
| Enzyme | Active site |
| HDAC4 | Zn2+ cofactor with Asp196, His198, and Asp290 residue | HDAC5 | Zn2+ cofactor with Asp870, His872, and Asp964 | HDAC6 | Zn2+ cofactor with Cys5, His7, and Cys78 | HDAC7 | Zn2+ cofactor with Asp707, His709, and Asp801 | HDAC9 | Zn2+ cofactor with Asp820, His822, and Asp914 | HDAC10 | Zn2+ cofactor with Asp172, His174, and Asp265 |
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