Research Article

Docking Studies and Biological Activity of Fosinopril Analogs

Table 2

Percent inhibition of ACE by A2 at different concentrations.

AnalogPercent inhibition
0.01 nM0.02 nM0.2 nM0.4 nM0.6 nM0.8 nM1 nM

A244.72 ± 3.8553.17 ± 5.7375.12 ± 4.6677.80 ± 3.2181.74 ± 6.0983.98 ± 5.1184.45 ± 4.52