Table 4: Oocyte electrophysiological data of benzodiazepines [87].

Compoundα1α2α3α5

SH-053-2′F-R-CH3 (2)111/154124/185125/220183/387
SH-053-2′F-S-CH3 (17)116/164170/348138/301218/389

Efficacy at αβ3γ2 receptor subtypes as % of control current at 100 nM and 1 μM concentrations. Data presented as percent over baseline (100) at concentrations of 100 nM/1 μM.