Review Article
Activators and Inhibitors of NRF2: A Review of Their Potential for Clinical Development
Table 2
Selected peptides acting as NRF2-KEAP1 protein-protein interaction inhibitors.
| Sequence | Mechanism of action | Reference |
| LDEETGEFL-NH2 | Binding to KEAP1-Kelch domain | [100, 101] | DEETGE-CAL-Tat (NH2-RKKRRQRRR-PLFAERLDEETGEFLPNH2) | [103] | Ac-DPETGEL-OH | [102] | FITCβ-DEETGEF-OH | [102] | FITC-β-LDEETGEFL-OH | [102] | Ac-DEETGEF-OH | [102] | Ac-DPETGEL-OH | [102] | FITC-LDEETGEFL-NH2 | [100] | FAM-LDEETGEFL-NH2 | [108] | LQLDEETGEFLPIQGK(MR121)-OH | [107] | Ac-LDEETGEFL-NH2 | [100, 101] | Ac-DPETGEL-NH2 | [104] | Ac-NPETGEL-OH | [104] | St-DPETGEL-OH | [104] | YGRKKRRQRRRLQLDEETGEFLPIQ | [162] | c[GQLDPETGEFL] | | [105] |
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