| Compounds | (IC50/EC50) µM |
| SCPIs | | N-(4-{[4-(3,4-Dichlorophenyl)-1,3-thiazol-2-yl]amino}phenyl)acetamidehydrobromide (SCPI-1) | 0.347 (IC50) | 8-Chloro-2-(3-methoxyphenyl)-4,4-dimethyl-4,5-dihydroisothiazolo[5,4-c]quinoline-1(2H)-thione (SCPI-2) | 0.059 (IC50) | 3-(4-Bromophenyl)-5-methoxy-7-nitro-4H-1,2,4-benzoxadiazine (SCPI-3) | 0.159 (IC50) | 4,4,8-Trimethyl-5-(3-methylbutanoyl)-4,5-dihydro-1H-[1,2]dithiolo[3,4-c]quinoline-1-thione (SCPI-4) | 0.065 (IC50) | 3-Bromo-N-{2-[(4-chloro-2-nitrophenyl)amino]ethyl}-4-ethoxybenzamide (SCPI-5) | 0.042 (IC50) |
| Synthetic analogs of curcumin | | (2E,6E)-2-6-Bis(3,4,5-trimethoxybenzylidene) cyclohexanone | 12.11 (EC50) | (2E,6E)-2-6-Bis(furan-2-ylmethylene) cyclohexanone | 62.87 (EC50) | (1E,4E)-1,5-Bis(4-hydroxyphenyl) penta-1,4-dien-3-one | 2.38 (EC50) | (1E,4E)-1-(2-Hydroxyphenyl)-5-phenylpenta-1,4-dien-3-one | 2.02 (EC50) | 1,5-Bis-(3,4,5-trimethoxy-phenyl)-penta-1,4-dien-3-one | 0.65 (EC50) |
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