Research Article

Compounds from Cynomorium songaricum with Estrogenic and Androgenic Activities Suppress the Oestrogen/Androgen-Induced BPH Process

Table 3

Summary of results on cellular level.

Number Abb. Androgenic activity Estrogen activity
AR
N.T.
AR
T.A.
LNCaP
Prol.
ERα
N.T.
ERα
T.A.
ERβ
N.T.
ERβ
T.A.
MCF7
Prol.

(1)FAN.D.+N.D.N.D.N.D.N.D.
(2)CynN.D.+N.D.N.D.N.D.N.D.
(3)UAN.D.+N.D.N.D.N.D.N.D.
(4)GalN.D.+N.D.N.D.N.D.N.D.
(5)PalN.D.+N.D.N.D.N.D.N.D.
(6)PacN.D.+N.D.N.D.N.D.N.D.
(7)Lut+N.D.+N.D.N.D.N.D.N.D.
(8)Rut+N.D.+N.D.N.D.N.D.N.D.
(9)ECG+++++N.D.++
(10)NarN.D.N.D.N.D.N.D.+N.D.++
(11)PhlN.D.N.D.N.D.N.D.+N.D.+
(12)ChrN.D.N.D.N.D.N.D.+N.D.+
(13)EmoN.D.N.D.N.D.N.D.+N.D.++
(14)PhyN.D.N.D.N.D.N.D.N.D.+
(15)CatN.D.N.D.N.D.N.D.N.D.

Note. “N.T.”: nuclear translocation, “T.A.”: transcriptional activity, “Prol.”: proliferation, “−”: negative, “+”: positive, and “N.D.”: has not been detected.