| Biological activity | Compounds | Reference |
| Anticancer | Isoliquiritigenin | [31–35] | Isoliquiritin | [32] | Licochalcone A | [36–42] | Licochalcone B | [43, 44] | Licochalcone C | [45, 46] | Licochalcone D | [45, 46] | Licochalcone E | [47–49] | Kanzonol C | [50] | Isobavachalcone | [51] | Echinatin | [52, 53] | Isoliquiritin apioside | [54] | Paratocarpin A | [55] | 4-Hydroxylonchocarpin | [56, 57] | Kanzonol Y | [58] |
| Anti-inflammatory | Isoliquiritin | [59] | Isoliquiritigenin | [59–68] | Homobutein | [68] | Echinatin | [10, 69, 70] | Licochalcone A | [10, 70–75] | Licochalcone B | [10, 21, 69, 70] | Licochalcone C | [21, 69, 76, 77] | Licochalcone D | [69, 70] | Licochalcone E | [21, 77] | Isobavachalcone | [78, 79] | Morachalcone A | [80] | Kanzonol B | [10, 79] | DTM | [10, 21] | Licoagrochalcone C | [10, 21] | 4-Hydroxylonchocarpin | [78, 81] |
| Antibacterial | Isoliquiritigenin | [82, 83] | Licochalcone A | [84–88] | Isobavachalcone | [89–91] | Kanzonol C | [89, 90] | 4-Hydroxylonchocarpin | [89] |
| Antiviral | Isoliquiritigenin | [28, 92] | Licochalcone A | [92, 93] | Isobavachalcone | [94] | Echinatin | [28] | Kanzonol Y | [95] |
| Antioxidative | Isoliquiritigenin | [26, 96] | Licochalcone A | [97, 98] | Licochalcone B | [10, 22] | Licochalcone C | [99] | Licochalcone D | [22] | Isobavachalcone | [100] | Echinatin | [10] | DTM | [10] | Paratocarpin B | [26] | Glypallichalcone | [101] | Dihydroisoliquiritigenin | [102] |
| Hepatoprotective | Isoliquiritigenin | [103] | Echinatin | [104] | Licochalcone A | [104] | Licochalcone B | [103–105] | Licochalcone E | [106] | Licoagrochalcone A | [103] | 3,4,3′,4′-Tetrahydroxychalcone | [103] |
| Antidiabetic | Isoliquiritigenin | [107, 108] | Licochalcone E | [12] | Echinatin | [109] | Isobavachalcone | [110] | Kanzonol C | [21] | Licoagrochalcone A | [21] |
| Antiobesity | Kanzonol C | [21] | Licoagrochalcone A | [21] | Isobavachalcone | [110] | Isoliquiritin apioside | [111] | Isoliquiritigenin | [111] | Licochalcone A | [112, 113] |
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