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S. No. | Patent application number | Year of filing | Applicant name | Patent office | Compound | Category |
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1 | AU 200521 958-B2 [6] | 2005 | Boehringer Ingelheim International GmbH | Australian | | DPP-IV inhibitor |
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2 | CA 02873524 [7] | 2007 | Boehringer Ingelheim International GmbH | Canadian | 1-[(4-methyl-quinazolin-2-yl)methyl]-3-7-(2-butyn-1-yl)-8-(3-(R)-aminopiperidin-1-yl) xanthine | DPP-IV inhibitor |
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3 | EP 2058311A2 [8] | 2003 | Boehringer Ingelheim International GmbH and Co. | European patent office | | DPP-IV inhibitor |
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4 | DE 6020050 00 986T2 [9] | 2005 | Loreal Paris | Deutsches patent under Markenamt | — | Obesity |
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5 | EP 1368349 B1 [10] | 2002 | Boehringer Ingelheim International GmbH and Co. | Europian | | DPP-IV |
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6 | EP 1515972 B1 [11] | 2003 | F.Hoffman-La Roche AG 4070 Basel (CH) | Europian | | Type-II diabetes |
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7 | EP 1599477 B1 [12] | 2004 | F.Hoffman-La Roche AG 4070 Basel (CH) | Europian | | PEPCK inhibitors |
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8 | EP 1689748 B1 [13] | 2004 | Boehringer Ingelheim International GmbH | Europian | | Diabetes |
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9 | ES 2401128 T3 [14] | 2006 | GlaxoSmithKline LLC | Spain | | Agonist of HM74 A |
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10 | US 7696212 B2 [15] | 2010 | Boehringer Ingelheim International GmbH and Co. KG | United States | | DPP-IV inhibitor |
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11 | US 7838529 B2 [16] | 2010 | Boehringer Ingelheim International GmbH, Ingelheimam Rhein (DE) | United States | | Type-2 diabetes mellitus, antiobesity. |
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12 | US 7879864 B2 [17] | 2011 | Sanofi-Aventis Deutschland GmbH, Frankfurt am main (DE) | United States | | DPP-IV inhibitor |
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13 | US 9221821 B2 [18] | 2015 | Forest Laboratories Holdings Limited, Hamilton (BM) | United States | | - |
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14 | US 10202383 B2 [19] | 2019 | Boehringer Ingelheim International GmbH, Ingelheim am Rhein (DE) | United States | | DPP-IV |
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15 | US 10214530 B2 [20] | 2019 | Max-Delbruck-Centrum Fur Molekulare Medizin, Berlin (De), Forschungs-Verbund-Berlin-E. V., Berlin (De) | United States | | Serotonin based disease |
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16 | US 201111 8464 [21] | 2009 | Ing-Jun Chen Linya District (TW) | United States | | Anticancer |
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