A Novel Nonpeptide CGRP Receptor Antagonist, ‘Compound 1’ (WO98/11128) Is a High Affinity Competitive Antagonist at the CGRP1 Receptor in Human Coronary Arteries
P. Hasbak,1,2O. Saetrum Opgaard,3K. Eskesen,1S. Schifter,2H. Arendrup,4J. Longmore,5and L. Edvinsson1